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Developmental Therapeutics Program (DTP)

Stage2 tested compounds

Inhibited Strains

NSC/name 1.2 microM 3.7 microM 11 microM 33 microM 100 microM Stage2 Graphs NCI 60 Human
Tumor Cell Data
3D Structure
of Compound
Basic Chemical Data
674565           Stage2 Graphs for 674565 60 Cell Data for 674565 3D Structure for 674565 Basic Chemical Data for 674565
674566           Stage2 Graphs for 674566 60 Cell Data for 674566 3D Structure for 674566 Basic Chemical Data for 674566
674573           Stage2 Graphs for 674573 60 Cell Data for 674573 3D Structure for 674573 Basic Chemical Data for 674573
674615         bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 674615 60 Cell Data for 674615 3D Structure for 674615 Basic Chemical Data for 674615
674699
9-[3-[N-(2-N,N-DIMETHYLAMINO)
ETHYL]AMINOPROPYL]AMINO-
1-NITROACRIDINE.3HCL
rad18 rad14 rad18 sgs1 rad14 rad18 rad52 sgs1 mec2 rad14 rad18 rad50 rad52 rad50EPP+ sgs1 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 rad50EPP+ sgs1 wt2 Stage2 Graphs for 674699 60 Cell Data for 674699 3D Structure for 674699 Basic Chemical Data for 674699
674709     wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 674709 60 Cell Data for 674709 3D Structure for 674709 Basic Chemical Data for 674709
674915       rad50EPP+ bub3 mec2 rad14 rad18 rad52 mgt1 mlh1 rad50EPP+ sgs1 Stage2 Graphs for 674915 60 Cell Data for 674915 3D Structure for 674915 Basic Chemical Data for 674915
675205       rad50 rad52 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 675205 60 Cell Data for 675205 3D Structure for 675205 Basic Chemical Data for 675205
675207         rad50 rad52 Stage2 Graphs for 675207 60 Cell Data for 675207 3D Structure for 675207 Basic Chemical Data for 675207
675209       rad50 rad52 rad50 rad52 Stage2 Graphs for 675209 60 Cell Data for 675209 3D Structure for 675209 Basic Chemical Data for 675209
675369         rad18 rad50 rad52 Stage2 Graphs for 675369 60 Cell Data for 675369 3D Structure for 675369 Basic Chemical Data for 675369
675583         mgt1 sgs1 Stage2 Graphs for 675583 60 Cell Data for 675583 3D Structure for 675583 Basic Chemical Data for 675583
676363
CYCLOBUTANEMETHANOL, 1-[[
(2,5-DIAMINO-4-CHLORO-6-
PYRIMIDINYL)AMINO]METHYL]- 3-
(2-PHENYLETHYL)-, DIHYDROCHLORIDE
      bub3 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 sgs1 Stage2 Graphs for 676363 60 Cell Data for 676363 3D Structure for 676363 Basic Chemical Data for 676363
676514
9-[3-(2-NITROAMIDAZOL-1-YL)
PROPYL]AMINO-1-NITROACRIDINE.HCL
rad18 rad14 rad18 sgs1 mec2 rad14 rad18 rad50 rad52 sgs1 CLN2oe mec2 rad14 rad18 rad50 rad52 mlh1 rad50EPP+ sgs1 wt2 all Stage2 Graphs for 676514 60 Cell Data for 676514 3D Structure for 676514 Basic Chemical Data for 676514
677395
2-AZIDO-10-[(4-DIMETHYLAMINO)
BUTYL]PHENOTHIAZINE,
OXALATE SALT
        all Stage2 Graphs for 677395 60 Cell Data for 677395 3D Structure for 677395 Basic Chemical Data for 677395
677438
ALDRITHIOL-2
    bub3 mec2 rad52 rad50EPP+ all all Stage2 Graphs for 677438   3D Structure for 677438 Basic Chemical Data for 677438
677450
2-AMINOPHENYL DISULFIDE
    bub3 mec2 mgt1 mlh1 rad50EPP+ sgs1 all CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 rad50EPP+ sgs1 wt2 Stage2 Graphs for 677450   3D Structure for 677450 Basic Chemical Data for 677450
677629
FURAN-2-CARBOXAMIDE, 3-(4-
CHLOROPHENYL)-N-CYCLOHEXYL
- 5-METHOXY-4-(PHENYLSULFONYL)-
    wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 677629 60 Cell Data for 677629 3D Structure for 677629 Basic Chemical Data for 677629
677936
ACETIC ACID, 2-[4-BROMO-5-(4-
BROMOPHENYL)-3-OXO- 2-
FURANYLIDENE]-, METHYL ESTER
      bub3 wt2 bub3 mec2 rad14 rad18 mgt1 rad50EPP+ wt2 Stage2 Graphs for 677936 60 Cell Data for 677936 3D Structure for 677936 Basic Chemical Data for 677936
678914
4-ACRIDINECARBOXAMIDE, N-
[2-(DIMETHYLAMINO)ETHYL]- 1-
METHOXY-, DIHYDROCHLORIDE
  rad50 rad50 rad52 rad50 rad52 rad50EPP+ CLN2oe mec2 rad50 rad52 mlh1 rad50EPP+ wt2 Stage2 Graphs for 678914 60 Cell Data for 678914 3D Structure for 678914 Basic Chemical Data for 678914
680418     mec2 sgs1 CLN2oe bub3 mec2 rad18 rad50 rad52 mgt1 mlh1 rad50EPP+ sgs1 wt2 all Stage2 Graphs for 680418 60 Cell Data for 680418 3D Structure for 680418 Basic Chemical Data for 680418
680434
3-AMINO-9-THIO-(10H)-ACRIDONE
        rad52 rad50EPP+ wt2 Stage2 Graphs for 680434 60 Cell Data for 680434 3D Structure for 680434 Basic Chemical Data for 680434
680510
1,8-NAPHTHYRIDIN-3-AMINE,
2,7-DICHLORO-5-METHYL-
        rad14 rad18 mgt1 mlh1 wt2 Stage2 Graphs for 680510 60 Cell Data for 680510 3D Structure for 680510 Basic Chemical Data for 680510
681286
9-CHLOR-2-METHYL-OXAZOLO
(4,5-C)QUINOLIN-4-ONE
        rad14 rad18 rad50 rad52 mgt1 mlh1 sgs1 Stage2 Graphs for 681286 60 Cell Data for 681286 3D Structure for 681286 Basic Chemical Data for 681286
681761     bub3 mec2 rad18 rad52 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 681761 60 Cell Data for 681761 3D Structure for 681761 Basic Chemical Data for 681761
681778       rad50EPP+ CLN2oe bub3 mec2 rad18 rad50 rad52 mgt1 mlh1 rad50EPP+ sgs1 wt2 Stage2 Graphs for 681778 60 Cell Data for 681778 3D Structure for 681778 Basic Chemical Data for 681778
682009       bub3 rad18 rad50 mgt1 mlh1 sgs1 wt2 bub3 mec2 rad18 rad52 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 682009 60 Cell Data for 682009 3D Structure for 682009 Basic Chemical Data for 682009
682127
BENZENE-1,3-BIS(ETHANEDI
THIOIC ACID), ALPHA,ALPHA'-
DIOXO-5-(1-OXOPROPYL)-,
DIMETHYL ESTER
    all all all Stage2 Graphs for 682127 60 Cell Data for 682127 3D Structure for 682127 Basic Chemical Data for 682127
682552         mec2 rad14 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 682552 60 Cell Data for 682552 3D Structure for 682552 Basic Chemical Data for 682552
682576     wt2 bub3 mec2 rad14 rad18 rad50 rad52 wt1 mlh1 sgs1 wt2 all Stage2 Graphs for 682576 60 Cell Data for 682576 3D Structure for 682576 Basic Chemical Data for 682576
682577     wt2 bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 rad50EPP+ sgs1 wt2 all Stage2 Graphs for 682577 60 Cell Data for 682577 3D Structure for 682577 Basic Chemical Data for 682577
683260   rad18 rad18 rad14 rad18 rad50EPP+ sgs1 all Stage2 Graphs for 683260 60 Cell Data for 683260 3D Structure for 683260 Basic Chemical Data for 683260
683414   rad50 rad52 rad50 rad52 rad50 rad52 CLN2oe mec2 rad50 rad52 Stage2 Graphs for 683414 60 Cell Data for 683414 3D Structure for 683414 Basic Chemical Data for 683414
683584         rad50 rad52 wt2 Stage2 Graphs for 683584 60 Cell Data for 683584 3D Structure for 683584 Basic Chemical Data for 683584
683591       CLN2oe bub3 mec2 rad18 rad50 rad52 mgt1 mlh1 wt2 all Stage2 Graphs for 683591 60 Cell Data for 683591 3D Structure for 683591 Basic Chemical Data for 683591
683635     CLN2oe bub3 rad18 rad50 rad52 mgt1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 683635 60 Cell Data for 683635 3D Structure for 683635 Basic Chemical Data for 683635
683792
4,4'-BIPIPERIDINE, 1,1'-BIS[(6-
METHOXY- 2-NAPHTHALENYL)
METHYL]-, DIHYDROCHLORIDE
        all Stage2 Graphs for 683792 60 Cell Data for 683792 3D Structure for 683792 Basic Chemical Data for 683792
683828     mgt1 bub3 rad14 mgt1 mlh1 wt2 bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 rad50EPP+ sgs1 wt2 Stage2 Graphs for 683828 60 Cell Data for 683828 3D Structure for 683828 Basic Chemical Data for 683828
683830           Stage2 Graphs for 683830 60 Cell Data for 683830 3D Structure for 683830 Basic Chemical Data for 683830
683831     all all all Stage2 Graphs for 683831 60 Cell Data for 683831 3D Structure for 683831 Basic Chemical Data for 683831
683863
HMAF
  rad18 rad18 rad18 rad18 rad50 rad52 sgs1 Stage2 Graphs for 683863 60 Cell Data for 683863 3D Structure for 683863 Basic Chemical Data for 683863
683909       CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 all Stage2 Graphs for 683909 60 Cell Data for 683909 3D Structure for 683909 Basic Chemical Data for 683909
683910       bub3 rad18 rad50 mgt1 sgs1 wt2 bub3 rad18 rad50 mgt1 sgs1 wt2 Stage2 Graphs for 683910 60 Cell Data for 683910 3D Structure for 683910 Basic Chemical Data for 683910
683919       CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 683919 60 Cell Data for 683919 3D Structure for 683919 Basic Chemical Data for 683919
684118
PYRIDO[3,4-G]QUINOLINE-5,10-
DIONE, 1,4-DIHYDRO- 1-(DI
METHYLAMINO)-4-METHYL-
  rad18 rad18 rad50 rad52 rad50EPP+ all all Stage2 Graphs for 684118 60 Cell Data for 684118 3D Structure for 684118 Basic Chemical Data for 684118
684405
1-(4'-PHTHALIMIDOPROPYL-
CARBONYL)-5-FLUOROURACIL
      mec2 mgt1 sgs1 mec2 rad50 mgt1 mlh1 rad50EPP+ sgs1 wt2 Stage2 Graphs for 684405 60 Cell Data for 684405 3D Structure for 684405 Basic Chemical Data for 684405
684839     CLN2oe bub3 mec2 rad52 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 684839 60 Cell Data for 684839 3D Structure for 684839 Basic Chemical Data for 684839
684853           Stage2 Graphs for 684853 60 Cell Data for 684853 3D Structure for 684853 Basic Chemical Data for 684853
684973       rad50EPP+ rad14 rad18 rad50 rad52 mgt1 mlh1 rad50EPP+ sgs1 wt2 Stage2 Graphs for 684973 60 Cell Data for 684973 3D Structure for 684973 Basic Chemical Data for 684973
684990       rad50EPP+ all Stage2 Graphs for 684990 60 Cell Data for 684990 3D Structure for 684990 Basic Chemical Data for 684990
685105
METHYL 4-[2-[4-BROMO-3,6-DIOXO
-1,4-CYCLOHEXADIENYL]
ETHYL]-BENZOATE
      wt2 rad52 rad50EPP+ wt2 Stage2 Graphs for 685105 60 Cell Data for 685105 3D Structure for 685105 Basic Chemical Data for 685105
685106
ISOPROPYL 4-[2-[4-BROMO-2,5-
DIHYDROXYPHENYL]ETHYL]
BENZOATE
  rad50EPP+ rad14 mgt1 mlh1 rad50EPP+ wt2 CLN2oe bub3 rad14 rad18 rad50 mgt1 mlh1 rad50EPP+ wt2 all Stage2 Graphs for 685106 60 Cell Data for 685106 3D Structure for 685106 Basic Chemical Data for 685106
685418         bub3 rad52 sgs1 wt2 Stage2 Graphs for 685418 60 Cell Data for 685418 3D Structure for 685418 Basic Chemical Data for 685418
685458           Stage2 Graphs for 685458 60 Cell Data for 685458 3D Structure for 685458 Basic Chemical Data for 685458
685529
LUPININE, O-METHOXYBENZOIC ACID
    rad14 mgt1 mlh1 rad50EPP+ wt2 bub3 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 rad50EPP+ wt2 all Stage2 Graphs for 685529 60 Cell Data for 685529 3D Structure for 685529 Basic Chemical Data for 685529
685922         rad50 rad52 sgs1 Stage2 Graphs for 685922 60 Cell Data for 685922 3D Structure for 685922 Basic Chemical Data for 685922
685967           Stage2 Graphs for 685967 60 Cell Data for 685967 3D Structure for 685967 Basic Chemical Data for 685967
686139           Stage2 Graphs for 686139 60 Cell Data for 686139 3D Structure for 686139 Basic Chemical Data for 686139
686315       CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 686315 60 Cell Data for 686315 3D Structure for 686315 Basic Chemical Data for 686315
686325   CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 all all Stage2 Graphs for 686325 60 Cell Data for 686325 3D Structure for 686325 Basic Chemical Data for 686325
686349
SPIRO[1,3-DITHIOLE-2,7'(3'H)-[1,2]
DITHIOLO[4,3-B]- THIOPYRAN]-4,5,5',6'-
TETRACARBOXYLIC ACID, 3'-OXO
  rad50 rad52 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 686349 60 Cell Data for 686349 3D Structure for 686349 Basic Chemical Data for 686349
686380       CLN2oe mec2 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 686380 60 Cell Data for 686380 3D Structure for 686380 Basic Chemical Data for 686380
686381       CLN2oe mec2 rad14 mgt1 mlh1 sgs1 wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 686381 60 Cell Data for 686381 3D Structure for 686381 Basic Chemical Data for 686381
686574
3H-1,2-BENZODITHIOL-3-ONE-1-
OXIDE
        bub3 mec2 rad18 rad50 rad52 mgt1 Stage2 Graphs for 686574 60 Cell Data for 686574 3D Structure for 686574 Basic Chemical Data for 686574
686612         sgs1 Stage2 Graphs for 686612 60 Cell Data for 686612 3D Structure for 686612 Basic Chemical Data for 686612
687330
ADENOSINE, 2'-AMINO-2'-DEOXY
-3',5'- O-[1,1,3,3-TETRAKIS(1-
METHYLETHYL)-1,3-DISILOXANEDIYL]
    wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 all Stage2 Graphs for 687330 60 Cell Data for 687330 3D Structure for 687330 Basic Chemical Data for 687330
687346       wt2 CLN2oe bub3 mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 687346 60 Cell Data for 687346 3D Structure for 687346 Basic Chemical Data for 687346
687355
1H-[1,2,4]TRIAZOLO[1,2-A]
PYRIDAZINE-8-CARBOXYLIC ACID,
5-[(2,3,4,6-O-TETRAACETYL-
BETA-D-GLUCOPYRAN
      wt2 CLN2oe bub3 rad18 rad52 sgs1 wt2 Stage2 Graphs for 687355 60 Cell Data for 687355 3D Structure for 687355 Basic Chemical Data for 687355
687370         rad18 rad50 mgt1 mlh1 sgs1 wt2 Stage2 Graphs for 687370 60 Cell Data for 687370 3D Structure for 687370 Basic Chemical Data for 687370
687605           Stage2 Graphs for 687605 60 Cell Data for 687605 3D Structure for 687605 Basic Chemical Data for 687605
687665       bub3 rad50EPP+ bub3 rad50EPP+ Stage2 Graphs for 687665 60 Cell Data for 687665 3D Structure for 687665 Basic Chemical Data for 687665
687666       rad50EPP+ rad50EPP+ Stage2 Graphs for 687666 60 Cell Data for 687666 3D Structure for 687666 Basic Chemical Data for 687666
687667     bub3 bub3 sgs1 bub3 mec2 rad14 rad18 rad50 rad52 mlh1 Stage2 Graphs for 687667 60 Cell Data for 687667 3D Structure for 687667 Basic Chemical Data for 687667
687668         bub3 Stage2 Graphs for 687668 60 Cell Data for 687668 3D Structure for 687668 Basic Chemical Data for 687668
687669         bub3 Stage2 Graphs for 687669 60 Cell Data for 687669 3D Structure for 687669 Basic Chemical Data for 687669
687670           Stage2 Graphs for 687670 60 Cell Data for 687670 3D Structure for 687670 Basic Chemical Data for 687670
687673       rad50EPP+ rad50EPP+ Stage2 Graphs for 687673 60 Cell Data for 687673 3D Structure for 687673 Basic Chemical Data for 687673
687826           Stage2 Graphs for 687826 60 Cell Data for 687826 3D Structure for 687826 Basic Chemical Data for 687826
688034
1-BUTYLOXYMETHYL-6-BROMO
-2,4(1H,3H)-QUINAZOLINEDIONE
          Stage2 Graphs for 688034 60 Cell Data for 688034 3D Structure for 688034 Basic Chemical Data for 688034
688036
3-BENZYLOXYMETHYL-4(3H)-
QUINAZALONE, HYDROCHLORIDE
          Stage2 Graphs for 688036 60 Cell Data for 688036 3D Structure for 688036 Basic Chemical Data for 688036
688114           Stage2 Graphs for 688114 60 Cell Data for 688114 3D Structure for 688114 Basic Chemical Data for 688114
688342           Stage2 Graphs for 688342 60 Cell Data for 688342 3D Structure for 688342 Basic Chemical Data for 688342
688484     mec2 rad14 rad18 rad50 rad52 wt1 mgt1 mlh1 rad50EPP+ sgs1 wt2 all all Stage2 Graphs for 688484 60 Cell Data for 688484 3D Structure for 688484 Basic Chemical Data for 688484
688542
5'-O-(DIMETHOXYTRITYL)-N(SUP
1)-(2-NITROBENZYL)-2-AZAINOSINE
          Stage2 Graphs for 688542 60 Cell Data for 688542 3D Structure for 688542 Basic Chemical Data for 688542
688791
BENZOIC ACID, 4-[[(3,6-DIOXO-
1,4-CYCLOHEXADIENYLMETHYL]
AMINO]-2-HYDROXY-, METHYL ESTER
    CLN2oe rad14 rad18 rad50 rad52 mgt1 mlh1 rad50EPP+ sgs1 wt2 all all Stage2 Graphs for 688791 60 Cell Data for 688791 3D Structure for 688791 Basic Chemical Data for 688791
689622       bub3 mec2 rad14 rad18 rad50 rad52 mgt1 mlh1 sgs1 rad14 rad18 rad50 mgt1 mlh1 Stage2 Graphs for 689622 60 Cell Data for 689622 3D Structure for 689622 Basic Chemical Data for 689622
689625         rad50EPP+ Stage2 Graphs for 689625 60 Cell Data for 689625 3D Structure for 689625 Basic Chemical Data for 689625
689626   rad50EPP+ rad50 rad52 rad50EPP+ CLN2oe bub3 mec2 rad18 rad50 rad52 wt1 mgt1 mlh1 rad50EPP+ sgs1 wt2 bub3 mec2 rad14 rad18 rad50 mgt1 mlh1 rad50EPP+ sgs1 Stage2 Graphs for 689626 60 Cell Data for 689626 3D Structure for 689626 Basic Chemical Data for 689626
709257
QUINOLINE, 7-CHLORO-4-[3-(2-
NITROIMIDAZOLYL)PROPYLAMINO
]-,HYDROCHLORIDE
          Stage2 Graphs for 709257 60 Cell Data for 709257 3D Structure for 709257 Basic Chemical Data for 709257