In Vivo Screening Data Summary

NCI In Vivo Screening Data

P388 Leukemia resistant to Tiazofurin; NSC 286193, Developed at LMCB,DTP,DCT,NCI (intraperitoneal) in CD2F1 (CDF1) mice

NSC 119875
CAS 15663-27-1
Cisplatin; Plantinol AQ; Cis-DDP

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX005 (ip) median survival time saline 0.38 mg/kg/injection 357.0 Antitumor endpoint evaluated on day 45; 06/06 animals surviving on day 5
Q01DX005 (ip) median survival time saline 0.38 mg/kg/injection 192.0 Antitumor endpoint evaluated on day 45; 06/06 animals surviving on day 5
Q01DX005 (ip) median survival time saline 0.75 mg/kg/injection 357.0 Antitumor endpoint evaluated on day 45; 06/06 animals surviving on day 5
Q01DX005 (ip) median survival time saline 0.75 mg/kg/injection 432.0 Antitumor endpoint evaluated on day 45; 06/06 animals surviving on day 5
Q01DX005 (ip) median survival time saline 1.5 mg/kg/injection 357.0 Antitumor endpoint evaluated on day 45; 06/06 animals surviving on day 5
Q01DX005 (ip) median survival time saline 1.5 mg/kg/injection 432.0 Antitumor endpoint evaluated on day 45; 06/06 animals surviving on day 5
Q01DX005 (ip) median survival time saline 3.0 mg/kg/injection 357.0 Antitumor endpoint evaluated on day 45; 05/06 animals surviving on day 5
Q01DX005 (ip) median survival time saline 3.0 mg/kg/injection 86.0 Antitumor endpoint evaluated on day 45; 06/06 animals surviving on day 5