In Vivo Screening Data Summary

NCI In Vivo Screening Data

B16 Melanoma (intraperitoneal) in BCF1 mice

NSC 119875
CAS 15663-27-1
Cisplatin; Plantinol AQ; Cis-DDP

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX009 (ip) median survival time saline 1.0 mg/kg/injection 137.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline 1.0 mg/kg/injection 155.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline 1.0 mg/kg/injection 179.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline 2.0 mg/kg/injection 152.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline 2.0 mg/kg/injection 178.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline 2.0 mg/kg/injection 194.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline 10.0 mg/kg/injection 157.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 9
Q01DX009 (ip) median survival time saline 10.0 mg/kg/injection 139.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 9
Q01DX009 (ip) median survival time saline 20.0 mg/kg/injection 141.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 9
Q01DX009 (ip) median survival time saline 20.0 mg/kg/injection 176.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 9