In Vivo Screening Data Summary

NCI In Vivo Screening Data

L1210 Leukemia resistant to BCNU; NSC 409962 (intraperitoneal) in B6D2F1 (BDF1) mice

NSC 119875
CAS 15663-27-1
Cisplatin; Plantinol AQ; Cis-DDP

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX005 (ip) mean survival time saline with Tween-80 2.7 mg/kg/injection 155.0 Antitumor endpoint evaluated on day 45; 09/10 animals surviving on tox evaluation day (usually day 5)
Q01DX005 (ip) mean survival time saline with Tween-80 4.0 mg/kg/injection 171.0 Antitumor endpoint evaluated on day 45; 09/10 animals surviving on tox evaluation day (usually day 5)
Q01DX005 (ip) mean survival time saline with Tween-80 6.0 mg/kg/injection 187.0 Antitumor endpoint evaluated on day 45; 10/10 animals surviving on tox evaluation day (usually day 5)
Q01DX005 (ip) mean survival time saline with Tween-80 9.0 mg/kg/injection 102.0 Antitumor endpoint evaluated on day 45; 10/10 animals surviving on tox evaluation day (usually day 5)