In Vivo Screening Data Summary

NCI In Vivo Screening Data

P388 Leukemia resistant to Cis DDPT; NSC 119875 (intraperitoneal) in B6D2F1 (BDF1) mice

NSC 119875
CAS 15663-27-1
Cisplatin; Plantinol AQ; Cis-DDP

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX001 (ip) median survival time saline 1.7 mg/kg/injection 108.0 Antitumor endpoint evaluated on day 30; 08/08 animals surviving on day 5
Q01DX001 (ip) median survival time saline 2.9 mg/kg/injection 122.0 Antitumor endpoint evaluated on day 30; 08/08 animals surviving on day 5
Q01DX001 (ip) median survival time saline 4.8 mg/kg/injection 127.0 Antitumor endpoint evaluated on day 30; 08/08 animals surviving on day 5
Q01DX001 (ip) median survival time saline 8.0 mg/kg/injection 142.0 Antitumor endpoint evaluated on day 30; 08/08 animals surviving on day 5
Q01DX001 (ip) median survival time saline 13.3 mg/kg/injection 143.0 Antitumor endpoint evaluated on day 30; 07/08 animals surviving on day 5