In Vivo Screening Data Summary

NCI In Vivo Screening Data

NCI-H23 Human Lung Adenocarcinoma (intrarenal inoculation) in NU/NU BALB/C (nude) mice

NSC 119875
CAS 15663-27-1
Cisplatin; Plantinol AQ; Cis-DDP

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q04DX004 (ip) mean tumor weight change saline 2.5 mg/kg/injection -53.0 Antitumor endpoint evaluated on day 18; 05/05 animals surviving on day 18
Q04DX004 (ip) mean tumor weight change saline 2.5 mg/kg/injection 2.0 Antitumor endpoint evaluated on day 18; 06/06 animals surviving on day 18
Q04DX004 (ip) mean tumor weight change saline 5.0 mg/kg/injection -88.0 Antitumor endpoint evaluated on day 18; 06/06 animals surviving on day 18
Q04DX004 (ip) mean tumor weight change saline 5.0 mg/kg/injection 2.0 Antitumor endpoint evaluated on day 18; 06/06 animals surviving on day 18
Q04DX004 (ip) mean tumor weight change saline 10.0 mg/kg/injection -98.0 Antitumor endpoint evaluated on day 18; 06/06 animals surviving on day 18
Q04DX004 (ip) mean tumor weight change saline 10.0 mg/kg/injection -66.0 Antitumor endpoint evaluated on day 18; 05/05 animals surviving on day 18
Q04DX004 (ip) mean tumor weight change saline 20.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 18; 01/06 animals surviving on day 18
Q04DX004 (ip) mean tumor weight change saline 20.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 18; 00/06 animals surviving on day 18