In Vivo Screening Data Summary

NCI In Vivo Screening Data

DU145 Human Prostate Tumor (intrarenal inoculation) in NU/NU BALB/C (nude) mice

NSC 119875
CAS 15663-27-1
Cisplatin; Plantinol AQ; Cis-DDP

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q04DX003 (ip) mean tumor weight change saline 2.5 mg/kg/injection 72.0 Antitumor endpoint evaluated on day 13; 06/06 animals surviving on day 13
Q04DX003 (ip) mean tumor weight change saline 2.5 mg/kg/injection 48.0 Antitumor endpoint evaluated on day 13; 06/06 animals surviving on day 13
Q04DX003 (ip) mean tumor weight change saline 5.0 mg/kg/injection 57.0 Antitumor endpoint evaluated on day 13; 06/06 animals surviving on day 13
Q04DX003 (ip) mean tumor weight change saline 5.0 mg/kg/injection 62.0 Antitumor endpoint evaluated on day 13; 06/06 animals surviving on day 13
Q04DX003 (ip) mean tumor weight change saline 10.0 mg/kg/injection 53.0 Antitumor endpoint evaluated on day 13; 06/06 animals surviving on day 13
Q04DX003 (ip) mean tumor weight change saline 10.0 mg/kg/injection 32.0 Antitumor endpoint evaluated on day 13; 06/06 animals surviving on day 13
Q04DX003 (ip) mean tumor weight change saline 20.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 13; 03/06 animals surviving on day 13
Q04DX003 (ip) mean tumor weight change saline 20.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 13; 02/06 animals surviving on day 13