In Vivo Screening Data Summary

NCI In Vivo Screening Data

L1210 Leukemia resistant to L-PAM; NSC 8806 (intraperitoneal) in CD2F1 (CDF1) mice

NSC 119875
CAS 15663-27-1
Cisplatin; Plantinol AQ; Cis-DDP

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX001 (ip) median survival time saline with Tween-80 5.3 mg/kg/injection 116.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX001 (ip) median survival time saline with Tween-80 5.3 mg/kg/injection 120.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX001 (ip) median survival time saline with Tween-80 8.0 mg/kg/injection 118.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX001 (ip) median survival time saline with Tween-80 8.0 mg/kg/injection 109.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX001 (ip) median survival time saline with Tween-80 10.0 mg/kg/injection 102.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX001 (ip) median survival time saline with Tween-80 10.0 mg/kg/injection 120.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 0.58 mg/kg/injection 107.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 0.58 mg/kg/injection 107.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 0.87 mg/kg/injection 110.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 0.87 mg/kg/injection 110.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 1.3 mg/kg/injection 128.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 1.3 mg/kg/injection 123.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 2.0 mg/kg/injection 119.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 2.0 mg/kg/injection 110.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5