In Vivo Screening Data Summary

NCI In Vivo Screening Data

P388 Leukemia resistant to AMSA; NSC 249992 (intraperitoneal) in CD2F1 (CDF1) mice

NSC 119875
CAS 15663-27-1
Cisplatin; Plantinol AQ; Cis-DDP

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q04DX003 (ip) median survival time saline 0.97 mg/kg/injection 182.0 Antitumor endpoint evaluated on day 45; 08/08 animals surviving on day 5
Q04DX003 (ip) median survival time saline 1.62 mg/kg/injection 208.0 Antitumor endpoint evaluated on day 45; 08/08 animals surviving on day 5
Q04DX003 (ip) median survival time saline 2.7 mg/kg/injection 295.0 Antitumor endpoint evaluated on day 45; 08/08 animals surviving on day 5
Q04DX003 (ip) median survival time saline 4.5 mg/kg/injection 391.0 Antitumor endpoint evaluated on day 45; 08/08 animals surviving on day 5
Q04DX003 (ip) median survival time saline 7.5 mg/kg/injection 230.0 Antitumor endpoint evaluated on day 45; 07/07 animals surviving on day 5