In Vivo Screening Data Summary

NCI In Vivo Screening Data

U-251 Human Glioma (intracerebral) in NU/NU BALB/C (nude) mice

NSC 119875
CAS 15663-27-1
Cisplatin; Plantinol AQ; Cis-DDP

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX005 (ip) median survival time saline 1.25 mg/kg/injection 93.0 Antitumor endpoint evaluated on day 75; 10/10 animals surviving on day 5
Q01DX005 (ip) median survival time saline 2.5 mg/kg/injection 97.0 Antitumor endpoint evaluated on day 75; 10/10 animals surviving on day 5
Q01DX005 (ip) median survival time saline 5.0 mg/kg/injection 137.0 Antitumor endpoint evaluated on day 75; 10/10 animals surviving on day 5
Q01DX005 (ip) median survival time saline 10.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 75; 09/10 animals surviving on day 5
Q01DX005 (ip) median survival time saline 20.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 75; 05/10 animals surviving on day 5