In Vivo Screening Data Summary

NCI In Vivo Screening Data

B16 Melanoma (intraperitoneal) in B6C3F1 mice

NSC 291305
CAS 1197-18-8
Tranexamic acid; DV79; DV 79

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX009 (ip) median survival time saline with Tween-80 12.5 mg/kg/injection 102.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 25.0 mg/kg/injection 101.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 50.0 mg/kg/injection 101.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 100.0 mg/kg/injection 101.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 200.0 mg/kg/injection 94.0 Antitumor endpoint evaluated on day 60; 09/10 animals surviving on day 5
Q01DX009 (ip) median survival time saline with Tween-80 400.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 60; 10/10 animals surviving on day 5