In Vivo Screening Data Summary

NCI In Vivo Screening Data

HT29;CX-1 Human Adenocarcinoma (MER+) (intrarenal inoculation) in NU/NU Swiss (nude) mice

NSC 291305
CAS 1197-18-8
Tranexamic acid; DV79; DV 79

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q04DX004 (sc) mean tumor weight change saline with Tween-80 200.0 mg/kg/injection 148.0 Antitumor endpoint evaluated on day 15; 06/06 animals surviving on day 15
Q04DX004 (sc) mean tumor weight change saline with Tween-80 400.0 mg/kg/injection 119.0 Antitumor endpoint evaluated on day 15; 06/06 animals surviving on day 15
Q04DX004 (sc) mean tumor weight change saline with Tween-80 800.0 mg/kg/injection 93.0 Antitumor endpoint evaluated on day 15; 06/06 animals surviving on day 15
Q04DX004 (sc) mean tumor weight change saline with Tween-80 1600.0 mg/kg/injection 112.0 Antitumor endpoint evaluated on day 15; 06/06 animals surviving on day 15