In Vivo Screening Data Summary

NCI In Vivo Screening Data

Colon Carcinoma 38 (subcutaneous) in B6D2F1 (BDF1) mice

NSC 291305
CAS 1197-18-8
Tranexamic acid; DV79; DV 79

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q07DX002 (ip) median tumor weight (est.) saline with Tween-80 25.0 mg/kg/injection 83.0 Antitumor endpoint evaluated on day 20; 10/10 animals surviving on day 20
Q07DX002 (ip) median tumor weight (est.) saline with Tween-80 50.0 mg/kg/injection 104.0 Antitumor endpoint evaluated on day 20; 10/10 animals surviving on day 20
Q07DX002 (ip) median tumor weight (est.) saline with Tween-80 100.0 mg/kg/injection 99.0 Antitumor endpoint evaluated on day 20; 10/10 animals surviving on day 20
Q07DX002 (ip) median tumor weight (est.) saline with Tween-80 200.0 mg/kg/injection 102.0 Antitumor endpoint evaluated on day 20; 10/10 animals surviving on day 20
Q07DX002 (ip) median tumor weight (est.) saline with Tween-80 400.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 20; 01/10 animals surviving on day 20
Q07DX002 (ip) median tumor weight (est.) saline with Tween-80 800.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 20; 00/10 animals surviving on day 20