In Vivo Screening Data Summary

NCI In Vivo Screening Data

Human Lung LX-1 Xenograft (intrarenal inoculation) in NU/NU Swiss (nude) mice

NSC 291305
CAS 1197-18-8
Tranexamic acid; DV79; DV 79

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q04DX003 (sc) mean tumor weight change saline with Tween-80 300.0 mg/kg/injection 167.0 Antitumor endpoint evaluated on day 11; 06/06 animals surviving on day 11
Q04DX003 (sc) mean tumor weight change saline with Tween-80 600.0 mg/kg/injection 104.0 Antitumor endpoint evaluated on day 11; 06/06 animals surviving on day 11
Q04DX003 (sc) mean tumor weight change saline with Tween-80 1200.0 mg/kg/injection 75.0 Antitumor endpoint evaluated on day 11; 06/06 animals surviving on day 11
Q04DX003 (sc) mean tumor weight change saline with Tween-80 2400.0 mg/kg/injection 79.0 Antitumor endpoint evaluated on day 11; 06/06 animals surviving on day 11