In Vivo Screening Data Summary

NCI In Vivo Screening Data

L1210 Leukemia (intraperitoneal) in B6D2F1 (BDF1) mice

NSC 97328
CAS 2208-07-3
EA hydrochloride; Ethyl acetimidate hydrochloride; Ethyl iminoacetate hydrochloride

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX001 (ip) mean survival time saline 50.0 mg/kg/injection 100.0 Antitumor endpoint evaluated on day 30; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX001 (ip) mean survival time saline 100.0 mg/kg/injection 89.0 Antitumor endpoint evaluated on day 30; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX001 (ip) mean survival time saline 200.0 mg/kg/injection 105.0 Antitumor endpoint evaluated on day 30; 06/06 animals surviving on tox evaluation day (usually day 5)
Q04DX003 (ip) mean survival time saline 100.0 mg/kg/injection 107.0 Antitumor endpoint evaluated on day 30; 03/03 animals surviving on tox evaluation day (usually day 5)
Q04DX003 (ip) mean survival time saline 200.0 mg/kg/injection 107.0 Antitumor endpoint evaluated on day 30; 03/03 animals surviving on tox evaluation day (usually day 5)
Q04DX003 (ip) mean survival time saline 400.0 mg/kg/injection 110.0 Antitumor endpoint evaluated on day 30; 03/03 animals surviving on tox evaluation day (usually day 5)