| Schedule (route) | Endpoint | Vehicle | Dose | Treated/Control (%) | Observations |
|---|---|---|---|---|---|
| Q01DX010 (ip) | mean tumor weight | other | 3.1 mg/kg/injection | 28.0 | Antitumor endpoint evaluated on day 21; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX010 (ip) | mean tumor weight | other | 6.2 mg/kg/injection | 16.0 | Antitumor endpoint evaluated on day 21; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX010 (ip) | mean tumor weight | other | 6.25 mg/kg/injection | 19.0 | Antitumor endpoint evaluated on day 21; 06/06 animals surviving on tox evaluation day (usually day 5) |
| Q01DX010 (ip) | mean tumor weight | other | 12.5 mg/kg/injection | 18.0 | Antitumor endpoint evaluated on day 21; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX010 (ip) | mean tumor weight | other | 25.0 mg/kg/injection | 9.0 | Antitumor endpoint evaluated on day 21; 05/06 animals surviving on tox evaluation day (usually day 5) |
| Q01DX010 (ip) | mean tumor weight | other | 25.0 mg/kg/injection | 10.0 | Antitumor endpoint evaluated on day 21; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX010 (ip) | mean tumor weight | other | 50.0 mg/kg/injection | 0.0 | Antitumor endpoint evaluated on day 21; 00/06 animals surviving on tox evaluation day (usually day 5) |
| Q01DX010 (ip) | mean tumor weight | other | 50.0 mg/kg/injection | 0.0 | Antitumor endpoint evaluated on day 21; 05/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX011 (ip) | mean tumor weight | other | 6.25 mg/kg/injection | 7.0 | Antitumor endpoint evaluated on day 21; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX011 (ip) | mean tumor weight | other | 12.5 mg/kg/injection | 4.0 | Antitumor endpoint evaluated on day 21; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX011 (ip) | mean tumor weight | other | 25.0 mg/kg/injection | 5.0 | Antitumor endpoint evaluated on day 21; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX011 (ip) | mean tumor weight | other | 50.0 mg/kg/injection | 7.0 | Antitumor endpoint evaluated on day 21; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX011 (ip) | mean tumor weight | other | 100.0 mg/kg/injection | 0.0 | Antitumor endpoint evaluated on day 14; 00/06 animals surviving on tox evaluation day (usually day 5) |
| Q01DX011 (ip) | mean tumor weight | other | 100.0 mg/kg/injection | 0.0 | Antitumor endpoint evaluated on day 21; 03/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX011 (ip) | mean tumor weight | other | 200.0 mg/kg/injection | 0.0 | Antitumor endpoint evaluated on day 14; 00/06 animals surviving on tox evaluation day (usually day 5) |