In Vivo Screening Data Summary

NCI In Vivo Screening Data

ADJ-PC-6 (intraperitoneal) in BALB/cJ mice

NSC 19893
CAS 51-21-8
Fluorouracil; Efudex; 5-FU

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q04DX003 (ip) median survival time saline 7.5 mg/kg/injection 471.0 Antitumor endpoint evaluated on day 90; 08/08 animals surviving on day 9
Q04DX003 (ip) median survival time saline 7.5 mg/kg/injection 150.0 Antitumor endpoint evaluated on day 60; 08/08 animals surviving on day 5
Q04DX003 (ip) median survival time saline 15.0 mg/kg/injection 308.0 Antitumor endpoint evaluated on day 90; 08/08 animals surviving on day 9
Q04DX003 (ip) median survival time saline 15.0 mg/kg/injection 173.0 Antitumor endpoint evaluated on day 60; 08/08 animals surviving on day 5
Q04DX003 (ip) median survival time saline 30.0 mg/kg/injection 471.0 Antitumor endpoint evaluated on day 90; 08/08 animals surviving on day 9
Q04DX003 (ip) median survival time saline 30.0 mg/kg/injection 150.0 Antitumor endpoint evaluated on day 75; 09/09 animals surviving on day 9
Q04DX003 (ip) median survival time saline 30.0 mg/kg/injection 273.0 Antitumor endpoint evaluated on day 60; 07/08 animals surviving on day 5
Q04DX003 (ip) median survival time saline 60.0 mg/kg/injection 471.0 Antitumor endpoint evaluated on day 90; 07/08 animals surviving on day 9
Q04DX003 (ip) median survival time saline 60.0 mg/kg/injection 193.0 Antitumor endpoint evaluated on day 75; 10/10 animals surviving on day 9
Q04DX003 (ip) median survival time saline 60.0 mg/kg/injection 335.0 Antitumor endpoint evaluated on day 60; 08/08 animals surviving on day 5
Q04DX003 (ip) median survival time saline 120.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 90; 05/08 animals surviving on day 9
Q04DX003 (ip) median survival time saline 120.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 75; 07/10 animals surviving on day 9
Q04DX003 (ip) median survival time saline 120.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 60; 08/08 animals surviving on day 5