In Vivo Screening Data Summary

NCI In Vivo Screening Data

L1210 Leukemia resistant to BCNU; NSC 409962 (subcutaneous) in B6D2F1 (BDF1) mice

NSC 755
CAS 50-44-2
Mercaptopurine; 6-Purinethiol; 6-Mercaptopurine

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX009 (ip) median survival time other 10.0 mg/kg/injection 122.0 Antitumor endpoint evaluated on day 38; 08/08 animals surviving on tox evaluation day (usually day 5)
Q01DX009 (ip) median survival time other 20.0 mg/kg/injection 133.0 Antitumor endpoint evaluated on day 38; 08/08 animals surviving on tox evaluation day (usually day 5)
Q01DX009 (ip) median survival time other 40.0 mg/kg/injection 161.0 Antitumor endpoint evaluated on day 38; 08/08 animals surviving on tox evaluation day (usually day 5)
Q01DX009 (ip) median survival time other 80.0 mg/kg/injection 155.0 Antitumor endpoint evaluated on day 38; 08/08 animals surviving on tox evaluation day (usually day 5)