| Schedule (route) | Endpoint | Vehicle | Dose | Treated/Control (%) | Observations |
|---|---|---|---|---|---|
| Q01DX009 (ip) | mean tumor weight | saline | 15.0 mg/kg/injection | 16.0 | Antitumor endpoint evaluated on day 28; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX009 (ip) | mean tumor weight | saline | 30.0 mg/kg/injection | 5.0 | Antitumor endpoint evaluated on day 28; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q01DX009 (ip) | mean tumor weight | saline | 60.0 mg/kg/injection | 14.0 | Antitumor endpoint evaluated on day 28; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | mean tumor weight | saline | 35.0 mg/kg/injection | 136.0 | Antitumor endpoint evaluated on day 33; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | mean tumor weight | saline | 67.5 mg/kg/injection | 57.0 | Antitumor endpoint evaluated on day 33; 09/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | mean tumor weight | saline | 135.0 mg/kg/injection | 37.0 | Antitumor endpoint evaluated on day 33; 07/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | saline | 4.0 mg/kg/injection | 73.0 | Antitumor endpoint evaluated on day 33; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | saline | 8.0 mg/kg/injection | 78.0 | Antitumor endpoint evaluated on day 33; 09/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | saline | 16.0 mg/kg/injection | 350.0 | Antitumor endpoint evaluated on day 33; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | saline | 32.0 mg/kg/injection | 78.0 | Antitumor endpoint evaluated on day 33; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | saline | 64.0 mg/kg/injection | 101.0 | Antitumor endpoint evaluated on day 33; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | saline | 128.0 mg/kg/injection | 28.0 | Antitumor endpoint evaluated on day 33; 08/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | Klucel (hydroxypropylcellulose) (HPC) | 6.25 mg/kg/injection | 78.0 | Antitumor endpoint evaluated on day 30; 09/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | Klucel (hydroxypropylcellulose) (HPC) | 12.5 mg/kg/injection | 131.0 | Antitumor endpoint evaluated on day 30; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | Klucel (hydroxypropylcellulose) (HPC) | 25.0 mg/kg/injection | 80.0 | Antitumor endpoint evaluated on day 30; 09/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | Klucel (hydroxypropylcellulose) (HPC) | 50.0 mg/kg/injection | 48.0 | Antitumor endpoint evaluated on day 30; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | median tumor weight (est.) | Klucel (hydroxypropylcellulose) (HPC) | 100.0 mg/kg/injection | 17.0 | Antitumor endpoint evaluated on day 30; 08/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | mean tumor weight (est.) | sodium bicarbonate | 67.5 mg/kg/injection | 136.0 | Antitumor endpoint evaluated on day 63; 08/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX005 (ip) | mean tumor weight (est.) | sodium bicarbonate | 135.0 mg/kg/injection | 42.0 | Antitumor endpoint evaluated on day 63; 04/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX006 (ip) | mean tumor weight | sodium bicarbonate | 67.5 mg/kg/injection | 49.0 | Antitumor endpoint evaluated on day 37; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX006 (ip) | mean tumor weight | sodium bicarbonate | 135.0 mg/kg/injection | 0.0 | Antitumor endpoint evaluated on day 37; 02/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX007 (ip) | mean tumor weight | saline | 35.0 mg/kg/injection | 98.0 | Antitumor endpoint evaluated on day 44; 10/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX007 (ip) | mean tumor weight | saline | 67.5 mg/kg/injection | 81.0 | Antitumor endpoint evaluated on day 44; 09/10 animals surviving on tox evaluation day (usually day 5) |
| Q07DX007 (ip) | mean tumor weight | saline | 135.0 mg/kg/injection | 0.0 | Antitumor endpoint evaluated on day 44; 06/10 animals surviving on tox evaluation day (usually day 5) |