In Vivo Screening Data Summary

NCI In Vivo Screening Data

Lymphosarcoma Gardner 6C3HED (intraperitoneal) in C3AKF1 (CHKRF1) mice

NSC 755
CAS 50-44-2
Mercaptopurine; 6-Purinethiol; 6-Mercaptopurine

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 5.0 mg/kg/injection 130.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 5.0 mg/kg/injection 130.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 5.0 mg/kg/injection 100.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 5.0 mg/kg/injection 108.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 10.0 mg/kg/injection 120.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 10.0 mg/kg/injection 104.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 10.0 mg/kg/injection 165.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 10.0 mg/kg/injection 108.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 20.0 mg/kg/injection 130.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 20.0 mg/kg/injection 100.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 20.0 mg/kg/injection 112.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 20.0 mg/kg/injection 115.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 40.0 mg/kg/injection 140.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 40.0 mg/kg/injection 100.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 40.0 mg/kg/injection 125.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 40.0 mg/kg/injection 130.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 80.0 mg/kg/injection 160.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 80.0 mg/kg/injection 129.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 80.0 mg/kg/injection 130.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)
Q01DX010 (ip) survival time, mean or median alkali diluted with saline 80.0 mg/kg/injection 120.0 Experiment continued until the death of all animals; 06/06 animals surviving on tox evaluation day (usually day 5)