In Vivo Screening Data Summary

NCI In Vivo Screening Data

HL-60 Human Promyelocytic Leukemia Xenograft (intraperitoneal) in NU/NU Swiss (nude) mice

NSC 19893
CAS 51-21-8
Fluorouracil; Efudex; 5-FU

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q04DX003 (ip) median survival time saline 50.0 mg/kg/injection 137.0 Antitumor endpoint evaluated on day 60; 08/08 animals surviving on day 9
Q04DX003 (ip) median survival time saline 75.0 mg/kg/injection 119.0 Antitumor endpoint evaluated on day 60; 07/08 animals surviving on day 9
Q04DX003 (ip) median survival time saline 112.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 60; 04/08 animals surviving on day 9