In Vivo Screening Data Summary

NCI In Vivo Screening Data

NCI-H125 Human Lung Adenosquamous Carcinoma (intrarenal inoculation) in NU/NU BALB/C (nude) mice

NSC 19893
CAS 51-21-8
Fluorouracil; Efudex; 5-FU

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q04DX003 (ip) mean tumor weight change saline 50.0 mg/kg/injection 60.0 Antitumor endpoint evaluated on day 16; 06/06 animals surviving on day 16
Q04DX003 (ip) mean tumor weight change saline 75.0 mg/kg/injection 62.0 Antitumor endpoint evaluated on day 16; 06/06 animals surviving on day 16
Q04DX003 (ip) mean tumor weight change saline 112.0 mg/kg/injection 66.0 Antitumor endpoint evaluated on day 16; 04/06 animals surviving on day 16