In Vivo Screening Data Summary

NCI In Vivo Screening Data

L1210 Leukemia resistant to Methane Sulfonate; NSC 102627 (intraperitoneal) in B6D2F1 (BDF1) mice

NSC 755
CAS 50-44-2
Mercaptopurine; 6-Purinethiol; 6-Mercaptopurine

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q01DX009 (ip) median survival time other 6.25 mg/kg/injection 97.0 Antitumor endpoint evaluated on day 30; 07/08 animals surviving on tox evaluation day (usually day 5)
Q01DX009 (ip) median survival time other 12.5 mg/kg/injection 101.0 Antitumor endpoint evaluated on day 30; 08/08 animals surviving on tox evaluation day (usually day 5)
Q01DX009 (ip) median survival time other 25.0 mg/kg/injection 103.0 Antitumor endpoint evaluated on day 30; 08/08 animals surviving on tox evaluation day (usually day 5)
Q01DX009 (ip) median survival time other 50.0 mg/kg/injection 124.0 Antitumor endpoint evaluated on day 30; 08/08 animals surviving on tox evaluation day (usually day 5)
Q01DX009 (ip) median survival time other 100.0 mg/kg/injection 86.0 Antitumor endpoint evaluated on day 30; 06/08 animals surviving on tox evaluation day (usually day 5)
Q01DX009 (ip) median survival time other 200.0 mg/kg/injection 87.0 Antitumor endpoint evaluated on day 30; 08/08 animals surviving on tox evaluation day (usually day 5)