In Vivo Screening Data Summary

NCI In Vivo Screening Data

Sarcoma M5076 (subcutaneous) in B6D2F1 (BDF1) mice

NSC 19893
CAS 51-21-8
Fluorouracil; Efudex; 5-FU

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q02DX033 (ip) median survival time saline 12.5 mg/kg/injection 101.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16
Q02DX033 (ip) median survival time saline 25.0 mg/kg/injection 105.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16
Q04DX006 (ip) median survival time saline 6.25 mg/kg/injection 105.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16
Q04DX006 (ip) median survival time saline 12.5 mg/kg/injection 100.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16
Q04DX006 (ip) median survival time saline 25.0 mg/kg/injection 108.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16
Q04DX006 (ip) median survival time saline 50.0 mg/kg/injection 105.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16