In Vivo Screening Data Summary

NCI In Vivo Screening Data

Sarcoma M5076 (subcutaneous) in B6D2F1 (BDF1) mice

NSC 755
CAS 50-44-2
Mercaptopurine; 6-Purinethiol; 6-Mercaptopurine

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q02DX033 (ip) median survival time saline with Tween-80 25.0 mg/kg/injection 0.0 Antitumor endpoint evaluated on day 100; 03/10 animals surviving on day 16
Q02DX033 (ip) median survival time saline with Tween-80 50.0 mg/kg/injection 107.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16
Q04DX006 (ip) median survival time saline with Tween-80 12.5 mg/kg/injection 99.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16
Q04DX006 (ip) median survival time saline with Tween-80 25.0 mg/kg/injection 111.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16
Q04DX006 (ip) median survival time saline with Tween-80 50.0 mg/kg/injection 105.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16
Q04DX006 (ip) median survival time saline with Tween-80 100.0 mg/kg/injection 111.0 Antitumor endpoint evaluated on day 100; 10/10 animals surviving on day 16