In Vivo Screening Data Summary

NCI In Vivo Screening Data

P388 Leukemia resistant to 5-Azacytidine; NSC 102816 (intraperitoneal) in CD2F1 (CDF1) mice

NSC 19893
CAS 51-21-8
Fluorouracil; Efudex; 5-FU

Chemical Data
Schedule (route) Endpoint Vehicle Dose Treated/Control (%) Observations
Q04DX002 (ip) median survival time saline 13.0 mg/kg/injection 147.0 Antitumor endpoint evaluated on day 35; 06/06 animals surviving on day 5
Q04DX002 (ip) median survival time saline 21.6 mg/kg/injection 156.0 Antitumor endpoint evaluated on day 35; 06/06 animals surviving on day 5
Q04DX002 (ip) median survival time saline 36.0 mg/kg/injection 164.0 Antitumor endpoint evaluated on day 35; 06/06 animals surviving on day 5
Q04DX002 (ip) median survival time saline 60.0 mg/kg/injection 173.0 Antitumor endpoint evaluated on day 35; 06/06 animals surviving on day 5
Q04DX002 (ip) median survival time saline 100.0 mg/kg/injection 194.0 Antitumor endpoint evaluated on day 35; 06/06 animals surviving on day 5